Browse by Authors and Editors
Number of items: 13.
Chen, Chou-Hsiung and Genapathy, Sivaneswary and Fischer, Peter M. and Chan, Weng C. (2014) A facile approach to tryptophan derivatives for the total synthesis of argyrin analogues. Organic and Biomolecular Chemistry, 12 (48). pp. 9764-9768. ISSN 1477-0539
Maryati, Marayti and Kaur, Ishwinder and Jadhav, Gopal P. and Olotu-Umoren, Loyin and Oveh, Blessing and Hashmi, Lubna and Fischer, Peter M. and Winkler, G. Sebastiaan (2013) A fluorescence-based assay suitable for quantitative analysis of deadenylase enzyme activity. Nucleic Acids Research . pp. 1-10. ISSN 0305-1048
Fischer, Peter M. (2017) Approved and experimental small-molecule oncology kinase inhibitor drugs: a mid-2016 overview. Medicinal Research Reviews, 37 (2). pp. 314-367. ISSN 1098-1128
Soukarieh, Fadi and Nowicki, Matthew W. and Bastide, Amandine and Poyry, Tuija and Jones, Carolyn and Dudek, Kate and Patwardhan, Geetanjali and Meullenet, François and Oldham, Neil J. and Walkinshaw, Malcolm D. and Willis, Anne E. and Fischer, Peter M. (2016) Design of nucleotide-mimetic and non-nucleotide inhibitors of the translation initiation factor eIF4E: synthesis, structural and functional characterisation. European Journal of Medicinal Chemistry, 124 . pp. 200-217. ISSN 0223-5234
Reddy, Tummala R.K. and Li, Chan and Guo, Xiaoxia and Fischer, Peter M. and Dekker, Lodewijk V. (2014) Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2–S100A10 protein interaction. Bioorganic and Medicinal Chemistry, 22 (19). pp. 5378-5391. ISSN 1464-3391
Zgair, Atheer and Wong, Jonathan C.M. and Lee, Jong Bong and Mistry, Jatin and Sivak, Olena and Wasan, Kishor M. and Hennig, Ivo M. and Barrett, David A. and Constantinescu, Cris S. and Fischer, Peter M. and Gershkovich, Pavel (2016) Dietary fats and pharmaceutical lipid excipients increase systemic exposure to orally administered cannabis and cannabis-based medicines. American Journal of Translational Research, 8 (8). pp. 3448-3459. ISSN 1943-8141
Emtage, Abigail L. and Mistry, Shailesh N. and Fischer, Peter M. and Kellam, Barrie and Laughton, Charles A. (2016) GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors. Journal of Biomolecular Structure and Dynamics . pp. 1-16. ISSN 1538-0254
Baker, Jillian G. and Mistry, Shailesh N. and Fischer, Peter M. and Hill, Stephen J. and Gardiner, Sheila M. and Kellam, Barrie (2012) In vitro and in vivo analysis of a novel highly selective β1-adrenoceptor partial agonist. In: British Pharmacological Society 4th Focused Meeting on Cell Signalling, 23-24 April 2012, Leicester, UK.
Baker, Jillian G. and Gardiner, Sheila M. and Woolard, Jeanette and Fromont, Christophe and Jadhav, Gopal P. and Mistry, Shailesh N. and Thompson, Kevin S.J. and Kellam, Barrie and Hill, Stephen J. and Fischer, Peter M. (2017) Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease. FASEB Journal . ISSN 1530-6860 (In Press)
Lee, Jong Bong and Zgair, Atheer and Taha, Dhiaa A. and Zang, Xiaowei and Kagan, Leonid and Kim, Tae Hwan and Kim, Min Gi and Yun, Hwi-yeol and Fischer, Peter M. and Gershkovich, Pavel (2017) Quantitative analysis of lab-to-lab variability in Caco-2 permeability assays. European Journal of Pharmaceutics and Biopharmaceutics . ISSN 1873-3441
Lee, Jong Bong and Zgair, Atheer and Kim, Tae Hwan and Kim, Min Gi and Yoo, Sun Dong and Fischer, Peter M. and Gershkovich, Pavel (2017) Simple and sensitive HPLC-UV method for determination of bexarotene in rat plasma. Journal of Chromatography B, 1040 . pp. 73-80. ISSN 1570-0232
Mistry, Shailesh Natvarbhai and Baker, Jillian G. and Fischer, Peter M. and Hill, Stephen J. and Gardiner, Sheila M. and Kellam, Barrie (2013) Synthesis and in vitro and in vivo characterization of highly β1-Selective β-Adrenoceptor partial agonists. Journal of Medicinal Chemistry, 56 (10). pp. 3852-3865. ISSN 0022-2623
Reddy, Tummala R.K. and Li, Chan and Fischer, Peter M. and Dekker, Lodewijk V. (2012) Three-dimensional pharmacophore design and biochemical screening identifies substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction. ChemMedChem, 7 (8). pp. 1435-1446. ISSN 1860-7179