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Lee, Jong Bong and Zgair, Atheer and Malec, Jed and Kim, Tae Hwan and Kim, Min Gi and Ali, Joseph and Qin, Chaolong and Feng, Wanshan and Chiang, Manting and Gao, Xizhe and Voronin, Gregory and Garces, Aimie and Lau, Chun Long and Chan, Ting-Hoi and Hume, Amy and McIntosh, Tecashanell M. and Soukarieh, Fadi and Al-Hayali, Mohammed and Cipolla, Elena and Collins, Hilary M. and Heery, David M. and Shin, Beom Soo and Yoo, Sun Dong and Kagan, Leonid and Stocks, Michael J. and Bradshaw, Tracey D. and Fischer, Peter M. and Gershkovich, Pavel (2018) Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system. Journal of Controlled Release, 286 . pp. 10-19. ISSN 1873-4995

Pearson, Russell J. and Blake, David G. and Mezna, Mokdad and Fischer, Peter M. and Westwood, Nicholas J. and McInnes, Campbell (2018) The Meisenheimer complex as a paradigm in drug discovery: reversible covalent inhibition through C67 of the ATP binding site of PLK1. Cell Chemical Biology . ISSN 2451-9456

Fridgeirsdottir, Gudrun and Harris, Robert and Dryden, Ian L. and Fischer, Peter M. and Roberts, Clive J. (2018) Multiple linear regression modelling to predict the stability of polymer-drug solid dispersions: comparison of the effects of polymers and manufacturing methods on solid dispersion stability. Molecular Pharmaceutics, 15 (5). pp. 1826-1841. ISSN 1543-8392

Zyryanova, Alisa F. and Weis, Félix and Faille, Alexandre and Abo Alard, Akeel and Crespillo-Casado, Ana and Sekine, Yusuke and Harding, Heather P. and Allen, Felicity and Parts, Leopold and Fromont, Christoph and Fischer, Peter M. and Warren, Alan J. and Ron, David (2018) Binding of ISRIB reveals a regulatory site in the nucleotide exchange factor eIF2B. Science, 359 (6383). pp. 1533-1536. ISSN 1095-9203

Whittaker, Steven R. and Barlow, Clare and Martin, Matthew P. and Mancusi, Caterina and Wagner, Steve and Self, Annette and Barrie, Elaine and te Poele, Robert and Sharp, Swee and Brown, Nathan and Wilson, Stuart and Jackson, Wayne and Fischer, Peter M. and Clarke, Paul A. and Walton, Michael I. and McDonald, Edward and Blagg, Julian and Noble, Martin and Garrett, Michelle D. and Workman, Paul (2018) Molecular profiling and combinatorial activity of CCT068127: a potent CDK2 and CDK9 inhibitor. Molecular Oncology, 12 (3). pp. 287-304. ISSN 1878-0261

Zgair, Atheer and Lee, Jong Bong and Wong, Jonathan Chi Man and Taha, Dhiaa A. and Aram, Jehan and Virgilio, Daisy Di and McArthur, Andrew G. and Cheng, Yu-Kit and Hennig, Ivo M. and Barrett, David A. and Fischer, Peter M. and Constantinescu, Cris S. and Gershkovich, Pavel (2017) Oral administration of cannabis with lipids leads to high levels of cannabinoids in the intestinal lymphatic system and prominent immunomodulation. Scientific Reports, 7 . 14542/1-14542/12. ISSN 2045-2322

Fischer, Peter M. (2017) Design of small-molecule active-site inhibitors of the S1A family proteases as procoagulant and anticoagulant drugs. Journal of Medicinal Chemistry, 61 (9). pp. 3799-3822. ISSN 1520-4804

Hamad, Badraldin K. and Pathak, Monika and Manna, Rosa and Fischer, Peter M. and Emsley, Jonas and Dekker, Lodewijk V. (2017) Assessment of the protein interaction between coagulation factor XII and corn trypsin inhibitor by molecular docking and biochemical validation. Journal of Thrombosis and Haemostasis, 15 (9). pp. 1818-1828. ISSN 1538-7836

Baker, Jillian G. and Gardiner, Sheila M. and Woolard, Jeanette and Fromont, Christophe and Jadhav, Gopal P. and Mistry, Shailesh N. and Thompson, Kevin S.J. and Kellam, Barrie and Hill, Stephen J. and Fischer, Peter M. (2017) Novel selective β1-adrenoceptor antagonists for concomitant cardiovascular and respiratory disease. FASEB Journal, 31 (7). pp. 3150-3166. ISSN 1530-6860

Lee, Jong Bong and Adrower, Cecilia and Qin, Chaolong and Fischer, Peter M. and Moor, Cornelia H. de and Gershkovich, Pavel (2017) Development of cordycepin formulations for preclinical and clinical studies. AAPS PharmSciTech . ISSN 1530-9932

Lee, Jong Bong and Zgair, Atheer and Taha, Dhiaa A. and Zang, Xiaowei and Kagan, Leonid and Kim, Tae Hwan and Kim, Min Gi and Yun, Hwi-yeol and Fischer, Peter M. and Gershkovich, Pavel (2017) Quantitative analysis of lab-to-lab variability in Caco-2 permeability assays. European Journal of Pharmaceutics and Biopharmaceutics, 114 . pp. 38-42. ISSN 1873-3441

Crespillo-Casado, Ana and Chambers, Joseph E. and Fischer, Peter M. and Marciniak, Stefan J. and Ron, David (2017) PPP1R15A-mediated dephosphorylation of eIF2α is unaffected by Sephin1 or Guanabenz. eLife, 6 . e26109/1-e26109/29. ISSN 2050-084X

Fischer, Peter M. (2017) Approved and experimental small-molecule oncology kinase inhibitor drugs: a mid-2016 overview. Medicinal Research Reviews, 37 (2). pp. 314-367. ISSN 1098-1128

Lee, Jong Bong and Zgair, Atheer and Kim, Tae Hwan and Kim, Min Gi and Yoo, Sun Dong and Fischer, Peter M. and Gershkovich, Pavel (2017) Simple and sensitive HPLC-UV method for determination of bexarotene in rat plasma. Journal of Chromatography B, 1040 . pp. 73-80. ISSN 1570-0232

Soukarieh, Fadi and Nowicki, Matthew W. and Bastide, Amandine and Poyry, Tuija and Jones, Carolyn and Dudek, Kate and Patwardhan, Geetanjali and Meullenet, François and Oldham, Neil J. and Walkinshaw, Malcolm D. and Willis, Anne E. and Fischer, Peter M. (2016) Design of nucleotide-mimetic and non-nucleotide inhibitors of the translation initiation factor eIF4E: synthesis, structural and functional characterisation. European Journal of Medicinal Chemistry, 124 . pp. 200-217. ISSN 0223-5234

Zgair, Atheer and Wong, Jonathan C.M. and Lee, Jong Bong and Mistry, Jatin and Sivak, Olena and Wasan, Kishor M. and Hennig, Ivo M. and Barrett, David A. and Constantinescu, Cris S. and Fischer, Peter M. and Gershkovich, Pavel (2016) Dietary fats and pharmaceutical lipid excipients increase systemic exposure to orally administered cannabis and cannabis-based medicines. American Journal of Translational Research, 8 (8). pp. 3448-3459. ISSN 1943-8141

Emtage, Abigail L. and Mistry, Shailesh N. and Fischer, Peter M. and Kellam, Barrie and Laughton, Charles A. (2016) GPCRs through the keyhole: the role of protein flexibility in ligand binding to β-adrenoceptors. Journal of Biomolecular Structure and Dynamics . pp. 1-16. ISSN 1538-0254

Chen, Chou-Hsiung and Genapathy, Sivaneswary and Fischer, Peter M. and Chan, Weng C. (2014) A facile approach to tryptophan derivatives for the total synthesis of argyrin analogues. Organic and Biomolecular Chemistry, 12 (48). pp. 9764-9768. ISSN 1477-0539

Reddy, Tummala R.K. and Li, Chan and Guo, Xiaoxia and Fischer, Peter M. and Dekker, Lodewijk V. (2014) Design, synthesis and SAR exploration of tri-substituted 1,2,4-triazoles as inhibitors of the annexin A2–S100A10 protein interaction. Bioorganic and Medicinal Chemistry, 22 (19). pp. 5378-5391. ISSN 1464-3391

Maryati, Marayti and Kaur, Ishwinder and Jadhav, Gopal P. and Olotu-Umoren, Loyin and Oveh, Blessing and Hashmi, Lubna and Fischer, Peter M. and Winkler, G. Sebastiaan (2013) A fluorescence-based assay suitable for quantitative analysis of deadenylase enzyme activity. Nucleic Acids Research . pp. 1-10. ISSN 0305-1048

Mistry, Shailesh N. and Baker, Jillian G. and Fischer, Peter M. and Hill, Stephen J. and Gardiner, Sheila M. and Kellam, Barrie (2013) Synthesis and in vitro and in vivo characterization of highly β1-Selective β-Adrenoceptor partial agonists. Journal of Medicinal Chemistry, 56 (10). pp. 3852-3865. ISSN 0022-2623

Reddy, Tummala R.K. and Li, Chan and Fischer, Peter M. and Dekker, Lodewijk V. (2012) Three-dimensional pharmacophore design and biochemical screening identifies substituted 1,2,4-triazoles as inhibitors of the annexin A2-S100A10 protein interaction. ChemMedChem, 7 (8). pp. 1435-1446. ISSN 1860-7179

Conference or Workshop Item

Baker, Jillian G. and Mistry, Shailesh N. and Fischer, Peter M. and Hill, Stephen J. and Gardiner, Sheila M. and Kellam, Barrie (2012) In vitro and in vivo analysis of a novel highly selective β1-adrenoceptor partial agonist. In: British Pharmacological Society 4th Focused Meeting on Cell Signalling, 23-24 April 2012, Leicester, UK.